| Entry ID |
Original Release date |
Data summary |
Entry Title |
Citation Title |
Authors |
| 53119 |
2026-01-06 |
Chemical Shifts: 1 set |
AR Tau-5* PP |
Oligomerization enables the selective targeting of an intrinsically disordered region by a small molecule
|
Antoni Riera, Borja Mateos, Carla Garcia-Cabau, Carolina Sanchez-Zarzalejo, Denes Hnisz, Henri Niskanen, Isabella C Felli, Jesus Garcia, Lorenzo Bracaglia, Marta Frigole-Vivas, Muhammad Awawdy, Roberta Pierattelli, Stase Bielskute, Xavier Salvatella |
| 53106 |
2026-01-06 |
Chemical Shifts: 1 set |
Androgen Receptor Tau-5* C404Y |
Oligomerization enables the selective targeting of an intrinsically disordered region by a small molecule
|
Antoni Riera, Borja Mateos, Carla Garcia-Cabau, Carolina Sanchez-Zarzalejo, Denes Hnisz, Henri Niskanen, Isabella C Felli, Jesus Garcia, Lorenzo Bracaglia, Marta Frigole-Vivas, Muhammad Awawdy, Roberta Pierattelli, Stase Bielskute, Xavier Salvatella |
| 53108 |
2026-01-06 |
Chemical Shifts: 1 set |
Androgen Receptor Nt L26P |
Oligomerization enables the selective targeting of an intrinsically disordered region by a small molecule
|
Antoni Riera, Borja Mateos, Carla Garcia-Cabau, Carolina Sanchez-Zarzalejo, Denes Hnisz, Henri Niskanen, Isabella C Felli, Jesus Garcia, Lorenzo Bracaglia, Marta Frigole-Vivas, Muhammad Awawdy, Roberta Pierattelli, Stase Bielskute, Xavier Salvatella |
| 53109 |
2026-01-06 |
Chemical Shifts: 1 set |
Androgen Receptor allTau-5 |
Oligomerization enables the selective targeting of an intrinsically disordered region by a small molecule
|
Antoni Riera, Borja Mateos, Carla Garcia-Cabau, Carolina Sanchez-Zarzalejo, Denes Hnisz, Henri Niskanen, Isabella C Felli, Jesus Garcia, Lorenzo Bracaglia, Marta Frigole-Vivas, Muhammad Awawdy, Roberta Pierattelli, Stase Bielskute, Xavier Salvatella |
| 53110 |
2026-01-12 |
Chemical Shifts: 1 set |
Androgen Receptor allTau-5 4G CtoS |
Oligomerization enables the selective targeting of an intrinsically disordered region by a small molecule
|
Antoni Riera, Borja Mateos, Carla Garcia-Cabau, Carolina Sanchez-Zarzalejo, Denes Hnisz, Henri Niskanen, Isabella C Felli, Jesus Garcia, Lorenzo Bracaglia, Marta Frigole-Vivas, Muhammad Awawdy, Roberta Pierattelli, Stase Bielskute, Xavier Salvatella |
| 53111 |
2026-01-12 |
Chemical Shifts: 1 set |
Androgen Receptor allTau-5 4G CtoS PP |
Oligomerization enables the selective targeting of an intrinsically disordered region by a small molecule
|
Antoni Riera, Borja Mateos, Carla Garcia-Cabau, Carolina Sanchez-Zarzalejo, Denes Hnisz, Henri Niskanen, Isabella C Felli, Jesus Garcia, Lorenzo Bracaglia, Marta Frigole-Vivas, Muhammad Awawdy, Roberta Pierattelli, Stase Bielskute, Xavier Salvatella |
| 53112 |
2026-01-06 |
Chemical Shifts: 1 set |
Progesterone Receptor Activation Domain (PR AD) |
Oligomerization enables the selective targeting of an intrinsically disordered region by a small molecule
|
Antoni Riera, Borja Mateos, Carla Garcia-Cabau, Carolina Sanchez-Zarzalejo, Denes Hnisz, Henri Niskanen, Isabella C Felli, Jesus Garcia, Lorenzo Bracaglia, Marta Frigole-Vivas, Muhammad Awawdy, Roberta Pierattelli, Stase Bielskute, Xavier Salvatella |
| 53113 |
2026-01-06 |
Chemical Shifts: 1 set |
AR Tau-5* C404S covalent dimer |
Oligomerization enables the selective targeting of an intrinsically disordered region by a small molecule
|
Antoni Riera, Borja Mateos, Carla Garcia-Cabau, Carolina Sanchez-Zarzalejo, Denes Hnisz, Henri Niskanen, Isabella C Felli, Jesus Garcia, Lorenzo Bracaglia, Marta Frigole-Vivas, Muhammad Awawdy, Roberta Pierattelli, Stase Bielskute, Xavier Salvatella |
| 53114 |
2026-01-06 |
Chemical Shifts: 1 set |
AR Tau-5* C404S C448-IAM |
Oligomerization enables the selective targeting of an intrinsically disordered region by a small molecule
|
Antoni Riera, Borja Mateos, Carla Garcia-Cabau, Carolina Sanchez-Zarzalejo, Denes Hnisz, Henri Niskanen, Isabella C Felli, Jesus Garcia, Lorenzo Bracaglia, Marta Frigole-Vivas, Muhammad Awawdy, Roberta Pierattelli, Stase Bielskute, Xavier Salvatella |
| 53115 |
2026-01-06 |
Chemical Shifts: 1 set |
AR Tau-5* (dC448) C404 - EPI-001 covalent adduct |
Oligomerization enables the selective targeting of an intrinsically disordered region by a small molecule
|
Antoni Riera, Borja Mateos, Carla Garcia-Cabau, Carolina Sanchez-Zarzalejo, Denes Hnisz, Henri Niskanen, Isabella C Felli, Jesus Garcia, Lorenzo Bracaglia, Marta Frigole-Vivas, Muhammad Awawdy, Roberta Pierattelli, Stase Bielskute, Xavier Salvatella |
| 53116 |
2026-01-06 |
Chemical Shifts: 1 set |
AR Tau-5* h2SA |
Oligomerization enables the selective targeting of an intrinsically disordered region by a small molecule
|
Antoni Riera, Borja Mateos, Carla Garcia-Cabau, Carolina Sanchez-Zarzalejo, Denes Hnisz, Henri Niskanen, Isabella C Felli, Jesus Garcia, Lorenzo Bracaglia, Marta Frigole-Vivas, Muhammad Awawdy, Roberta Pierattelli, Stase Bielskute, Xavier Salvatella |
| 53117 |
2026-01-06 |
Chemical Shifts: 1 set |
AR Tau-5* h3A |
Oligomerization enables the selective targeting of an intrinsically disordered region by a small molecule
|
Antoni Riera, Borja Mateos, Carla Garcia-Cabau, Carolina Sanchez-Zarzalejo, Denes Hnisz, Henri Niskanen, Isabella C Felli, Jesus Garcia, Lorenzo Bracaglia, Marta Frigole-Vivas, Muhammad Awawdy, Roberta Pierattelli, Stase Bielskute, Xavier Salvatella |
| 53118 |
2026-01-06 |
Chemical Shifts: 1 set |
AR Tau-5* L436P |
Oligomerization enables the selective targeting of an intrinsically disordered region by a small molecule
|
Antoni Riera, Borja Mateos, Carla Garcia-Cabau, Carolina Sanchez-Zarzalejo, Denes Hnisz, Henri Niskanen, Isabella C Felli, Jesus Garcia, Lorenzo Bracaglia, Marta Frigole-Vivas, Muhammad Awawdy, Roberta Pierattelli, Stase Bielskute, Xavier Salvatella |
| 53096 |
2026-01-07 |
Chemical Shifts: 1 set |
Estrogen Receptor alpha Activation Domain (ERa AD) |
Oligomerization enables the selective targeting of an intrinsically disordered region by a small molecule
|
Antoni Riera, Borja Mateos, Carla Garcia-Cabau, Carolina Sanchez-Zarzalejo, Denes Hnisz, Henri Niskanen, Isabella C Felli, Jesus Garcia, Lorenzo Bracaglia, Marta Frigole-Vivas, Muhammad Awawdy, Roberta Pierattelli, Stase Bielskute, Xavier Salvatella |
| 53097 |
2026-01-06 |
Chemical Shifts: 1 set |
Glucocorticoid receptor Activation Domain (GR AD) |
Oligomerization enables the selective targeting of an intrinsically disordered region by a small molecule
|
Antoni Riera, Borja Mateos, Carla Garcia-Cabau, Carolina Sanchez-Zarzalejo, Denes Hnisz, Henri Niskanen, Isabella C Felli, Jesus Garcia, Lorenzo Bracaglia, Marta Frigole-Vivas, Muhammad Awawdy, Roberta Pierattelli, Stase Bielskute, Xavier Salvatella |
| 53098 |
2026-01-06 |
Chemical Shifts: 1 set |
Mineralocorticoid Receptor Activation Domain (MR AD) |
Oligomerization enables the selective targeting of an intrinsically disordered region by a small molecule
|
Antoni Riera, Borja Mateos, Carla Garcia-Cabau, Carolina Sanchez-Zarzalejo, Denes Hnisz, Henri Niskanen, Isabella C Felli, Jesus Garcia, Lorenzo Bracaglia, Marta Frigole-Vivas, Muhammad Awawdy, Roberta Pierattelli, Stase Bielskute, Xavier Salvatella |
| 53099 |
2026-01-06 |
Chemical Shifts: 1 set |
Mineralocorticoid Receptor Activation Domain (MR AD) 2M urea |
Oligomerization enables the selective targeting of an intrinsically disordered region by a small molecule
|
Antoni Riera, Borja Mateos, Carla Garcia-Cabau, Carolina Sanchez-Zarzalejo, Denes Hnisz, Henri Niskanen, Isabella C Felli, Jesus Garcia, Lorenzo Bracaglia, Marta Frigole-Vivas, Muhammad Awawdy, Roberta Pierattelli, Stase Bielskute, Xavier Salvatella |
| 53100 |
2026-01-12 |
Chemical Shifts: 1 set |
Androgen Receptor Tau-5* noAro |
Oligomerization enables the selective targeting of an intrinsically disordered region by a small molecule
|
Antoni Riera, Borja Mateos, Carla Garcia-Cabau, Carolina Sanchez-Zarzalejo, Denes Hnisz, Henri Niskanen, Isabella C Felli, Jesus Garcia, Lorenzo Bracaglia, Marta Frigole-Vivas, Muhammad Awawdy, Roberta Pierattelli, Stase Bielskute, Xavier Salvatella |
| 53101 |
2026-01-06 |
Chemical Shifts: 1 set |
Androgen Receptor Tau-5* A398P |
Oligomerization enables the selective targeting of an intrinsically disordered region by a small molecule
|
Antoni Riera, Borja Mateos, Carla Garcia-Cabau, Carolina Sanchez-Zarzalejo, Denes Hnisz, Henri Niskanen, Isabella C Felli, Jesus Garcia, Lorenzo Bracaglia, Marta Frigole-Vivas, Muhammad Awawdy, Roberta Pierattelli, Stase Bielskute, Xavier Salvatella |
| 53102 |
2026-01-06 |
Chemical Shifts: 1 set |
Androgen Receptor Tau-5* AAA |
Oligomerization enables the selective targeting of an intrinsically disordered region by a small molecule
|
Antoni Riera, Borja Mateos, Carla Garcia-Cabau, Carolina Sanchez-Zarzalejo, Denes Hnisz, Henri Niskanen, Isabella C Felli, Jesus Garcia, Lorenzo Bracaglia, Marta Frigole-Vivas, Muhammad Awawdy, Roberta Pierattelli, Stase Bielskute, Xavier Salvatella |
| 53103 |
2026-01-06 |
Chemical Shifts: 1 set |
Androgen Receptor Tau-5* G407A |
Oligomerization enables the selective targeting of an intrinsically disordered region by a small molecule
|
Antoni Riera, Borja Mateos, Carla Garcia-Cabau, Carolina Sanchez-Zarzalejo, Denes Hnisz, Henri Niskanen, Isabella C Felli, Jesus Garcia, Lorenzo Bracaglia, Marta Frigole-Vivas, Muhammad Awawdy, Roberta Pierattelli, Stase Bielskute, Xavier Salvatella |
| 53104 |
2026-01-07 |
Chemical Shifts: 1 set |
Androgen Receptor Tau-5* dC448 |
Oligomerization enables the selective targeting of an intrinsically disordered region by a small molecule
|
Antoni Riera, Borja Mateos, Carla Garcia-Cabau, Carolina Sanchez-Zarzalejo, Denes Hnisz, Henri Niskanen, Isabella C Felli, Jesus Garcia, Lorenzo Bracaglia, Marta Frigole-Vivas, Muhammad Awawdy, Roberta Pierattelli, Stase Bielskute, Xavier Salvatella |
| 53105 |
2026-01-06 |
Chemical Shifts: 1 set |
Androgen Receptor Tau-5* |
Oligomerization enables the selective targeting of an intrinsically disordered region by a small molecule
|
Antoni Riera, Borja Mateos, Carla Garcia-Cabau, Carolina Sanchez-Zarzalejo, Denes Hnisz, Henri Niskanen, Isabella C Felli, Jesus Garcia, Lorenzo Bracaglia, Marta Frigole-Vivas, Muhammad Awawdy, Roberta Pierattelli, Stase Bielskute, Xavier Salvatella |
| 51479 |
2022-09-30 |
Chemical Shifts: 1 set |
Androgen Receptor AF1star |
Rational optimization of a transcription factor activation domain inhibitor
|
Albert Escobedo, Alessandro Ruffoni, Antoni Riera, Borja Mateos, C Adriana A Banuelos, Carla Garcia-Cabau, Carolina Sanchez-Zarzalejo, Cristina Batlle, David Meierhofer, Denes Hnisz, Elzbieta Szulc, Hannes Dockx, Harpreet Kaur, Isabelle Brun-Heath, Jesus Garcia, Jiaqi Zhu, Jon K Obst, Jordann Smak, Jun Wang, Karina Pombo-Garcia, Levente Zodi, Lidia Bardia, Marianne D Sadar, Marta Frigole-Vivas, Mateusz Biesaga, Michael Lewis, Mireia Pesarrodona, Nasrin R Mawji, Paula Martinez-Cristobal, Paul Robustelli, Salvador Ventura, Shaon Basu, Stase Bielskute, Teresa Tam, Travis H Stracker, Xavier Salvatella, Xavier Verdaguer |
| 51480 |
2023-11-17 |
Chemical Shifts: 1 set |
Androgen Receptor NTD |
Rational optimization of a transcription factor activation domain inhibitor
|
Albert Escobedo, Alessandro Ruffoni, Antoni Riera, Borja Mateos, C Adriana A Banuelos, Carla Garcia-Cabau, Carolina Sanchez-Zarzalejo, Cristina Batlle, David Meierhofer, Denes Hnisz, Elzbieta Szulc, Hannes Dockx, Harpreet Kaur, Isabelle Brun-Heath, Jesus Garcia, Jiaqi Zhu, Jon K Obst, Jordann Smak, Jun Wang, Karina Pombo-Garcia, Levente Zodi, Lidia Bardia, Marianne D Sadar, Marta Frigole-Vivas, Mateusz Biesaga, Michael Lewis, Mireia Pesarrodona, Nasrin R Mawji, Paula Martinez-Cristobal, Paul Robustelli, Salvador Ventura, Shaon Basu, Stase Bielskute, Teresa Tam, Travis H Stracker, Xavier Salvatella, Xavier Verdaguer |
| 51476 |
2023-11-17 |
Chemical Shifts: 1 set |
Androgen Receptor C-terminal NTD |
Rational optimization of a transcription factor activation domain inhibitor
|
Albert Escobedo, Alessandro Ruffoni, Antoni Riera, Borja Mateos, C Adriana A Banuelos, Carla Garcia-Cabau, Carolina Sanchez-Zarzalejo, Cristina Batlle, David Meierhofer, Denes Hnisz, Elzbieta Szulc, Hannes Dockx, Harpreet Kaur, Isabelle Brun-Heath, Jesus Garcia, Jiaqi Zhu, Jon K Obst, Jordann Smak, Jun Wang, Karina Pombo-Garcia, Levente Zodi, Lidia Bardia, Marianne D Sadar, Marta Frigole-Vivas, Mateusz Biesaga, Michael Lewis, Mireia Pesarrodona, Nasrin R Mawji, Paula Martinez-Cristobal, Paul Robustelli, Salvador Ventura, Shaon Basu, Stase Bielskute, Teresa Tam, Travis H Stracker, Xavier Salvatella, Xavier Verdaguer |
| 34491 |
2021-01-26 |
Chemical Shifts: 1 set |
Cortistatin analog with improved immunoregulatory activity |
Structure-based design of a Cortistatin analogue with immunomodulatory activity in models of inflammatory bowel disease
|
A Escola, A Riera, A Rol, B Ponsati, E Aragon, E Gonzalez-Rey, E Puig, J Farrera-Sinfreu, J Fernandez-Carneado, M Delgado, M J Macias, M Valles-Miret, P Martin-Malpartida, T Todorovski, X Verdaguer |
| 27548 |
2018-11-15 |
Chemical Shifts: 1 set |
Ressonance assignments for the human Smad5 MH1 domain |
TGIF1 homeodomain interacts with Smad MH1 domain and represses TGF-beta signaling.
|
Agnieszka Konkol, Antoni Riera, Carles Torner, David Sunol, Eric Aragon, Ewelina Guca, Jorge Cordero, Lidia Ruiz, Maria J Macias, Pau Martin-Malpartida |
| 27461 |
2018-07-17 |
Chemical Shifts: 1 set |
Human TGIF1 c-term domain |
TGIF1 homeodomain interacts with Smad MH1 domain and represses TGF-beta signaling.
|
Agnieszka Konkol, Antoni Riera, Carles Torner, David Sunol, Eric Aragon, Ewelina Guca, Jorge Cordero, Lidia Ruiz, Maria J Macias, Pau Martin-Malpartida |
| 26794 |
2016-08-31 |
Chemical Shifts: 1 set |
NMR Assignment of L-Dfp6,D-Trp8-SRIF |
Peptide aromatic interactions modulated by fluorinated residues: Synthesis, structure and biological activity of Somatostatin analogs containing 3-(3',5'difluorophenyl)-alanine
|
Alvaro Rol, Antoni Riera, Berta Ponsati, Eric Aragon, Jimena Fernandez-Carneado, Maria J Macias, Mariona Valles-Miret, Pablo Martin-Gago, Pau Martin-Malpartida, Toni Todorovski, Xavier Verdaguer |
| 26796 |
2016-08-31 |
Chemical Shifts: 1 set |
NMR Assignment of L-Dfp11,D-Trp8-SRIF |
Peptide aromatic interactions modulated by fluorinated residues: Synthesis, structure and biological activity of Somatostatin analogs containing 3-(3',5'difluorophenyl)-alanine
|
Alvaro Rol, Antoni Riera, Berta Ponsati, Eric Aragon, Jimena Fernandez-Carneado, Maria J Macias, Mariona Valles-Miret, Pablo Martin-Gago, Pau Martin-Malpartida, Toni Todorovski, Xavier Verdaguer |
| 26797 |
2016-08-31 |
Chemical Shifts: 1 set |
NMR Assignment of L-Dfp6,L-Msa7,D-Trp8-SRIF |
Peptide aromatic interactions modulated by fluorinated residues: Synthesis, structure and biological activity of Somatostatin analogs containing 3-(3',5'difluorophenyl)-alanine
|
Alvaro Rol, Antoni Riera, Berta Ponsati, Eric Aragon, Jimena Fernandez-Carneado, Maria J Macias, Mariona Valles-Miret, Pablo Martin-Gago, Pau Martin-Malpartida, Toni Todorovski, Xavier Verdaguer |
| 26798 |
2016-08-31 |
Chemical Shifts: 1 set |
NMR Assignment of L-Dfp11,L-Msa7,D-Trp8-SRIF |
Peptide aromatic interactions modulated by fluorinated residues: Synthesis, structure and biological activity of Somatostatin analogs containing 3-(3',5'difluorophenyl)-alanine
|
Alvaro Rol, Antoni Riera, Berta Ponsati, Eric Aragon, Jimena Fernandez-Carneado, Maria J Macias, Mariona Valles-Miret, Pablo Martin-Gago, Pau Martin-Malpartida, Toni Todorovski, Xavier Verdaguer |
| 26799 |
2016-08-31 |
Chemical Shifts: 1 set |
NMR Assignment of L-Dfp6,L-Msa7,D-Trp8, L-Dfp11-SRIF |
Peptide aromatic interactions modulated by fluorinated residues: Synthesis, structure and biological activity of Somatostatin analogs containing 3-(3',5'difluorophenyl)-alanine
|
Alvaro Rol, Antoni Riera, Berta Ponsati, Eric Aragon, Jimena Fernandez-Carneado, Maria J Macias, Mariona Valles-Miret, Pablo Martin-Gago, Pau Martin-Malpartida, Toni Todorovski, Xavier Verdaguer |
| 26795 |
2016-08-31 |
Chemical Shifts: 1 set |
NMR Assignment of L-Dfp7,D-Trp8-SRIF |
Peptide aromatic interactions modulated by fluorinated residues: Synthesis, structure and biological activity of Somatostatin analogs containing 3-(3',5'difluorophenyl)-alanine
|
Alvaro Rol, Antoni Riera, Berta Ponsati, Eric Aragon, Jimena Fernandez-Carneado, Maria J Macias, Mariona Valles-Miret, Pablo Martin-Gago, Pau Martin-Malpartida, Toni Todorovski, Xavier Verdaguer |