| Entry ID |
Original Release date |
Data summary |
Entry Title |
Citation Title |
Authors |
| 53119 |
2026-01-06 |
Chemical Shifts: 1 set |
AR Tau-5* PP |
Oligomerization enables the selective targeting of an intrinsically disordered region by a small molecule
|
Antoni Riera, Borja Mateos, Carla Garcia-Cabau, Carolina Sanchez-Zarzalejo, Denes Hnisz, Henri Niskanen, Isabella C Felli, Jesus Garcia, Lorenzo Bracaglia, Marta Frigole-Vivas, Muhammad Awawdy, Roberta Pierattelli, Stase Bielskute, Xavier Salvatella |
| 53116 |
2026-01-06 |
Chemical Shifts: 1 set |
AR Tau-5* h2SA |
Oligomerization enables the selective targeting of an intrinsically disordered region by a small molecule
|
Antoni Riera, Borja Mateos, Carla Garcia-Cabau, Carolina Sanchez-Zarzalejo, Denes Hnisz, Henri Niskanen, Isabella C Felli, Jesus Garcia, Lorenzo Bracaglia, Marta Frigole-Vivas, Muhammad Awawdy, Roberta Pierattelli, Stase Bielskute, Xavier Salvatella |
| 53117 |
2026-01-06 |
Chemical Shifts: 1 set |
AR Tau-5* h3A |
Oligomerization enables the selective targeting of an intrinsically disordered region by a small molecule
|
Antoni Riera, Borja Mateos, Carla Garcia-Cabau, Carolina Sanchez-Zarzalejo, Denes Hnisz, Henri Niskanen, Isabella C Felli, Jesus Garcia, Lorenzo Bracaglia, Marta Frigole-Vivas, Muhammad Awawdy, Roberta Pierattelli, Stase Bielskute, Xavier Salvatella |
| 53118 |
2026-01-06 |
Chemical Shifts: 1 set |
AR Tau-5* L436P |
Oligomerization enables the selective targeting of an intrinsically disordered region by a small molecule
|
Antoni Riera, Borja Mateos, Carla Garcia-Cabau, Carolina Sanchez-Zarzalejo, Denes Hnisz, Henri Niskanen, Isabella C Felli, Jesus Garcia, Lorenzo Bracaglia, Marta Frigole-Vivas, Muhammad Awawdy, Roberta Pierattelli, Stase Bielskute, Xavier Salvatella |
| 53097 |
2026-01-06 |
Chemical Shifts: 1 set |
Glucocorticoid receptor Activation Domain (GR AD) |
Oligomerization enables the selective targeting of an intrinsically disordered region by a small molecule
|
Antoni Riera, Borja Mateos, Carla Garcia-Cabau, Carolina Sanchez-Zarzalejo, Denes Hnisz, Henri Niskanen, Isabella C Felli, Jesus Garcia, Lorenzo Bracaglia, Marta Frigole-Vivas, Muhammad Awawdy, Roberta Pierattelli, Stase Bielskute, Xavier Salvatella |
| 53098 |
2026-01-06 |
Chemical Shifts: 1 set |
Mineralocorticoid Receptor Activation Domain (MR AD) |
Oligomerization enables the selective targeting of an intrinsically disordered region by a small molecule
|
Antoni Riera, Borja Mateos, Carla Garcia-Cabau, Carolina Sanchez-Zarzalejo, Denes Hnisz, Henri Niskanen, Isabella C Felli, Jesus Garcia, Lorenzo Bracaglia, Marta Frigole-Vivas, Muhammad Awawdy, Roberta Pierattelli, Stase Bielskute, Xavier Salvatella |
| 53099 |
2026-01-06 |
Chemical Shifts: 1 set |
Mineralocorticoid Receptor Activation Domain (MR AD) 2M urea |
Oligomerization enables the selective targeting of an intrinsically disordered region by a small molecule
|
Antoni Riera, Borja Mateos, Carla Garcia-Cabau, Carolina Sanchez-Zarzalejo, Denes Hnisz, Henri Niskanen, Isabella C Felli, Jesus Garcia, Lorenzo Bracaglia, Marta Frigole-Vivas, Muhammad Awawdy, Roberta Pierattelli, Stase Bielskute, Xavier Salvatella |
| 53101 |
2026-01-06 |
Chemical Shifts: 1 set |
Androgen Receptor Tau-5* A398P |
Oligomerization enables the selective targeting of an intrinsically disordered region by a small molecule
|
Antoni Riera, Borja Mateos, Carla Garcia-Cabau, Carolina Sanchez-Zarzalejo, Denes Hnisz, Henri Niskanen, Isabella C Felli, Jesus Garcia, Lorenzo Bracaglia, Marta Frigole-Vivas, Muhammad Awawdy, Roberta Pierattelli, Stase Bielskute, Xavier Salvatella |
| 53102 |
2026-01-06 |
Chemical Shifts: 1 set |
Androgen Receptor Tau-5* AAA |
Oligomerization enables the selective targeting of an intrinsically disordered region by a small molecule
|
Antoni Riera, Borja Mateos, Carla Garcia-Cabau, Carolina Sanchez-Zarzalejo, Denes Hnisz, Henri Niskanen, Isabella C Felli, Jesus Garcia, Lorenzo Bracaglia, Marta Frigole-Vivas, Muhammad Awawdy, Roberta Pierattelli, Stase Bielskute, Xavier Salvatella |
| 53103 |
2026-01-06 |
Chemical Shifts: 1 set |
Androgen Receptor Tau-5* G407A |
Oligomerization enables the selective targeting of an intrinsically disordered region by a small molecule
|
Antoni Riera, Borja Mateos, Carla Garcia-Cabau, Carolina Sanchez-Zarzalejo, Denes Hnisz, Henri Niskanen, Isabella C Felli, Jesus Garcia, Lorenzo Bracaglia, Marta Frigole-Vivas, Muhammad Awawdy, Roberta Pierattelli, Stase Bielskute, Xavier Salvatella |
| 53105 |
2026-01-06 |
Chemical Shifts: 1 set |
Androgen Receptor Tau-5* |
Oligomerization enables the selective targeting of an intrinsically disordered region by a small molecule
|
Antoni Riera, Borja Mateos, Carla Garcia-Cabau, Carolina Sanchez-Zarzalejo, Denes Hnisz, Henri Niskanen, Isabella C Felli, Jesus Garcia, Lorenzo Bracaglia, Marta Frigole-Vivas, Muhammad Awawdy, Roberta Pierattelli, Stase Bielskute, Xavier Salvatella |
| 53106 |
2026-01-06 |
Chemical Shifts: 1 set |
Androgen Receptor Tau-5* C404Y |
Oligomerization enables the selective targeting of an intrinsically disordered region by a small molecule
|
Antoni Riera, Borja Mateos, Carla Garcia-Cabau, Carolina Sanchez-Zarzalejo, Denes Hnisz, Henri Niskanen, Isabella C Felli, Jesus Garcia, Lorenzo Bracaglia, Marta Frigole-Vivas, Muhammad Awawdy, Roberta Pierattelli, Stase Bielskute, Xavier Salvatella |
| 53108 |
2026-01-06 |
Chemical Shifts: 1 set |
Androgen Receptor Nt L26P |
Oligomerization enables the selective targeting of an intrinsically disordered region by a small molecule
|
Antoni Riera, Borja Mateos, Carla Garcia-Cabau, Carolina Sanchez-Zarzalejo, Denes Hnisz, Henri Niskanen, Isabella C Felli, Jesus Garcia, Lorenzo Bracaglia, Marta Frigole-Vivas, Muhammad Awawdy, Roberta Pierattelli, Stase Bielskute, Xavier Salvatella |
| 53109 |
2026-01-06 |
Chemical Shifts: 1 set |
Androgen Receptor allTau-5 |
Oligomerization enables the selective targeting of an intrinsically disordered region by a small molecule
|
Antoni Riera, Borja Mateos, Carla Garcia-Cabau, Carolina Sanchez-Zarzalejo, Denes Hnisz, Henri Niskanen, Isabella C Felli, Jesus Garcia, Lorenzo Bracaglia, Marta Frigole-Vivas, Muhammad Awawdy, Roberta Pierattelli, Stase Bielskute, Xavier Salvatella |
| 53112 |
2026-01-06 |
Chemical Shifts: 1 set |
Progesterone Receptor Activation Domain (PR AD) |
Oligomerization enables the selective targeting of an intrinsically disordered region by a small molecule
|
Antoni Riera, Borja Mateos, Carla Garcia-Cabau, Carolina Sanchez-Zarzalejo, Denes Hnisz, Henri Niskanen, Isabella C Felli, Jesus Garcia, Lorenzo Bracaglia, Marta Frigole-Vivas, Muhammad Awawdy, Roberta Pierattelli, Stase Bielskute, Xavier Salvatella |
| 53113 |
2026-01-06 |
Chemical Shifts: 1 set |
AR Tau-5* C404S covalent dimer |
Oligomerization enables the selective targeting of an intrinsically disordered region by a small molecule
|
Antoni Riera, Borja Mateos, Carla Garcia-Cabau, Carolina Sanchez-Zarzalejo, Denes Hnisz, Henri Niskanen, Isabella C Felli, Jesus Garcia, Lorenzo Bracaglia, Marta Frigole-Vivas, Muhammad Awawdy, Roberta Pierattelli, Stase Bielskute, Xavier Salvatella |
| 53114 |
2026-01-06 |
Chemical Shifts: 1 set |
AR Tau-5* C404S C448-IAM |
Oligomerization enables the selective targeting of an intrinsically disordered region by a small molecule
|
Antoni Riera, Borja Mateos, Carla Garcia-Cabau, Carolina Sanchez-Zarzalejo, Denes Hnisz, Henri Niskanen, Isabella C Felli, Jesus Garcia, Lorenzo Bracaglia, Marta Frigole-Vivas, Muhammad Awawdy, Roberta Pierattelli, Stase Bielskute, Xavier Salvatella |
| 53115 |
2026-01-06 |
Chemical Shifts: 1 set |
AR Tau-5* (dC448) C404 - EPI-001 covalent adduct |
Oligomerization enables the selective targeting of an intrinsically disordered region by a small molecule
|
Antoni Riera, Borja Mateos, Carla Garcia-Cabau, Carolina Sanchez-Zarzalejo, Denes Hnisz, Henri Niskanen, Isabella C Felli, Jesus Garcia, Lorenzo Bracaglia, Marta Frigole-Vivas, Muhammad Awawdy, Roberta Pierattelli, Stase Bielskute, Xavier Salvatella |
| 51479 |
2022-09-30 |
Chemical Shifts: 1 set |
Androgen Receptor AF1star |
Rational optimization of a transcription factor activation domain inhibitor
|
Albert Escobedo, Alessandro Ruffoni, Antoni Riera, Borja Mateos, C Adriana A Banuelos, Carla Garcia-Cabau, Carolina Sanchez-Zarzalejo, Cristina Batlle, David Meierhofer, Denes Hnisz, Elzbieta Szulc, Hannes Dockx, Harpreet Kaur, Isabelle Brun-Heath, Jesus Garcia, Jiaqi Zhu, Jon K Obst, Jordann Smak, Jun Wang, Karina Pombo-Garcia, Levente Zodi, Lidia Bardia, Marianne D Sadar, Marta Frigole-Vivas, Mateusz Biesaga, Michael Lewis, Mireia Pesarrodona, Nasrin R Mawji, Paula Martinez-Cristobal, Paul Robustelli, Salvador Ventura, Shaon Basu, Stase Bielskute, Teresa Tam, Travis H Stracker, Xavier Salvatella, Xavier Verdaguer |
| 51480 |
2023-11-17 |
Chemical Shifts: 1 set |
Androgen Receptor NTD |
Rational optimization of a transcription factor activation domain inhibitor
|
Albert Escobedo, Alessandro Ruffoni, Antoni Riera, Borja Mateos, C Adriana A Banuelos, Carla Garcia-Cabau, Carolina Sanchez-Zarzalejo, Cristina Batlle, David Meierhofer, Denes Hnisz, Elzbieta Szulc, Hannes Dockx, Harpreet Kaur, Isabelle Brun-Heath, Jesus Garcia, Jiaqi Zhu, Jon K Obst, Jordann Smak, Jun Wang, Karina Pombo-Garcia, Levente Zodi, Lidia Bardia, Marianne D Sadar, Marta Frigole-Vivas, Mateusz Biesaga, Michael Lewis, Mireia Pesarrodona, Nasrin R Mawji, Paula Martinez-Cristobal, Paul Robustelli, Salvador Ventura, Shaon Basu, Stase Bielskute, Teresa Tam, Travis H Stracker, Xavier Salvatella, Xavier Verdaguer |
| 51476 |
2023-11-17 |
Chemical Shifts: 1 set |
Androgen Receptor C-terminal NTD |
Rational optimization of a transcription factor activation domain inhibitor
|
Albert Escobedo, Alessandro Ruffoni, Antoni Riera, Borja Mateos, C Adriana A Banuelos, Carla Garcia-Cabau, Carolina Sanchez-Zarzalejo, Cristina Batlle, David Meierhofer, Denes Hnisz, Elzbieta Szulc, Hannes Dockx, Harpreet Kaur, Isabelle Brun-Heath, Jesus Garcia, Jiaqi Zhu, Jon K Obst, Jordann Smak, Jun Wang, Karina Pombo-Garcia, Levente Zodi, Lidia Bardia, Marianne D Sadar, Marta Frigole-Vivas, Mateusz Biesaga, Michael Lewis, Mireia Pesarrodona, Nasrin R Mawji, Paula Martinez-Cristobal, Paul Robustelli, Salvador Ventura, Shaon Basu, Stase Bielskute, Teresa Tam, Travis H Stracker, Xavier Salvatella, Xavier Verdaguer |